1. Imvelaphi yezityalo kunye nokuSetyenziswa kweSintu
Igqabi le-Mulberry (Morus alba L.) liqulethe:
1-Deoxynojirimycin (DNJ)(0.1{1}}0.3%) - Enamandla -glucosidase inhibitor
IiFlavonoids(i-quercetin, isoquerctrin)
Iipolyphenols(i-chlorogenic acid, irutin)
Iirekhodi zembali:
Isishwankathelo seMateria Medica sichaza iimpawu zayo ezichasayo-sesifo seswekile
IsiNtu saseJapani "seswekile{0}}iti yothintelo"
2. Amacandelo angundoqo kunye neeNdlela zokuSebenza
2.1 Ulawulo lweGlucose Metabolism

2.2 Ii-Bioactives kunye neeThagethi
|
Icandelo |
Umxholo |
Ekujoliswe kuko |
Isiphumo |
|
1-Deoxynojirimycin |
0.1-0.3% |
Umda webrashi yamathumbu |
Yehlisa ukufunxwa kweglucose |
|
I-Quercetin-3-glucoside |
1.2-2.5% |
Indlela ye-AMPK |
Iphucula ubuntununtunu kwi-insulin |
|
I-Chlorogenic acid |
0.8-1.5% |
PPAR ukumodareyitha |
Inqanda i-gluconeogenesis yesibindi |
3. IMigangatho yoMgangatho
3.1 Uqinisekiso
Imicroscope: Iimpawu ezingezizo{0}}inwele zedlala ezidumbileyo
Iminwe ye-TLC: Kufuneka iindawo ezi-5 ezahlukeneyo
Ubungakanani beHPLC: Enkulu kuno okanye ilingana ne 0.1% DNJ (Pharmacopoeia standard)
3.2 IiNgcaciso zale mihla
I-Pharmacopoeia yaseTshayina: Iyonke i-flavonoids Enkulu okanye ilingana ne-1.5%
Umgangatho waseJapan: DNJ Inkulu kune okanye ilingana ne-0.15%
Ummiselo we-EU: iintsalela zezitshabalalisi<0.01ppm
4. Ubungqina beklinikhi
4.1 Ulawulo lwesifo seswekile
Uhlobo lwe-II DM: I-1200mg / ngosuku inciphisa i-HbA1c ngo-0.8-1.2%
I-Prediabetes: NNT =8 ukunqanda ukuqhubeka kwesifo seswekile
4.2 Izibonelelo zeMetabolic
Ukulawulwa kweLipid: 15-20% yokunciphisa i-triglyceride
Ulawulo lobunzima: 2-3cm esinqeni ukuncipha (iiveki ezili-12)
5. USebenziso lokuSebenzisa
5.1 ISicwangciso sokuThatha
Isiseko: 300mg (30min phambi{2}}isidlo)
Inzulu: 600mg + chromium combo
5.2 IiNdibaniselwano zeSynergistic
Gymnema sylvestre: Yongeza ukukhutshwa kwe-insulin
Alpha -lipoic acid: Ukuphucula ukusetyenziswa kwe-glucose ye-peripheral
Iiprobiotics: Ihlengahlengisa amathumbu -i-pancreas axis
6. Iingqwalasela zoKhuseleko
Umngcipheko we-Hypoglycemia: Ifuna esweni nge-antidiabetics
Izigulana zotyando: Susa iveki e-1 phambi{1}}phambi
GI ubuntununtunu: Qala ngeedosi eziphantsi
7. Isikhokelo sokuKhethwa kweMveliso
Umboniso weeMveliso zePremium:
Ibhalwe umxholo we-DNJ
Utsalo{0}}lobushushu obuphantsi
Iingxelo zovavanyo lwentsimbi enzima
Imiba eqhelekileyo:
Ukutshintshwa ngeentlobo ezisezantsi{0}}zeDNJ
Ukukrexeza kweDNJ yokwenziwa
8. Imida yoPhando
Amathumbu microbiota: Yandisa Akkermansia ubuninzi
Ukuphuculwa kwe-NAFLD: Ithintela iiseli ze-hepatic stellate
{0}}Izilungiso ezizisiweyo: Yandisa umsebenzi we-DNJ
Isiphelo sezeNzululwazi
Isicatshulwa samagqabi e-Mulberry sihambisa:
1️⃣ Multi{0}}ummiselo ojolise kuko(ithumbu+isibindi+izihlunu zeperipheral)
2️⃣ Ukhuseleko lwendalo(Imbali yokusetyenziswa kweminyaka engama-2000)
3️⃣ Iinzuzo ezibanzi zemetabolism(iglucose+lipids+ubunzima)




